Covalent inhibitors: a rational approach to drug discovery
Copyright policy )EC| AEGIS ,
EC| PROMINENT ,
NIH| Real-time discovery of inhibitors among billion compounds for preview and download ,
EC| EUC²LID
Fandi Sutanto; Markella Konstantinidou; Alexander Dömling;
Covalent inhibitors: a rational approach to drug discovery
In this review we provide a brief historic overview of covalent inhibitors and summarize recent advances focusing on developments in the last decade. Applications in challenging targets and future perspectives are also discussed.
Netherlands
- ACADEMISCH ZIEKENHUIS GRONINGEN Netherlands
- University of Gronigen Netherlands
- University of Groningen; Department of Pharmacy Netherlands
- University of Groningen Netherlands
Chemistry, POTENT
Chemistry, POTENT
citations This is an alternative to the "Influence" indicator, which also reflects the overall/total impact of an article in the research community at large, based on the underlying citation network (diachronically).222 popularity This indicator reflects the "current" impact/attention (the "hype") of an article in the research community at large, based on the underlying citation network.Top 0.1% influence This indicator reflects the overall/total impact of an article in the research community at large, based on the underlying citation network (diachronically).Top 10% impulse This indicator reflects the initial momentum of an article directly after its publication, based on the underlying citation network.Top 0.1%
citations
Citations provided by BIP!
This is an alternative to the "Influence" indicator, which also reflects the overall/total impact of an article in the research community at large, based on the underlying citation network (diachronically).
Citations provided by BIP!popularityPopularity provided by BIP!
This indicator reflects the "current" impact/attention (the "hype") of an article in the research community at large, based on the underlying citation network.
Popularity provided by BIP! 222
Top 0.1%
Top 10%
Top 0.1%
Green
hybrid
