BindingDB Entry 50028591: The discovery of potent, selective, and orally bioavailable PDE9 inhibitors as potential hypoglycemic agents.

Name: BindingDB Entry 50028591: The discovery of potent, selective, and orally bioavailable PDE9 inhibitors as potential hypoglycemic agents.
Creator: BindingDB

Research datakeyboard_double_arrow_right Dataset 01 Jan 2010 English Publisher:BindingDB

Authors: BindingDB;

doi: 10.7270/q2rb74gg

BindingDB Entry 50028591: The discovery of potent, selective, and orally bioavailable PDE9 inhibitors as potential hypoglycemic agents.

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Abstract

Small molecule binding data for protein Phosphodiesterase 1, Phosphodiesterase 1A (PDE1A), Phosphodiesterase 1C (PDE1C), Phosphodiesterase 3 (PDE3), Phosphodiesterase 7, Phosphodiesterase 8, cAMP-specific 3',5'-cyclic phosphodiesterase 4A, cAMP-specific 3',5'-cyclic phosphodiesterase 4B, cAMP-specific 3',5'-cyclic phosphodiesterase 4C, cAMP-specific 3',5'-cyclic phosphodiesterase 4D, cAMP-specific 3',5'-cyclic phosphodiesterase 7B, cGMP-inhibited 3',5'-cyclic phosphodiesterase B, and cGMP-specific 3',5'-cyclic phosphodiesterase, Uniprot O60658, O76074, O95263, P27815, P54750, Q01064, Q07343, Q08493, Q08499, Q13370, Q13946, Q14123, Q14432, and Q9NP56

Keywords

Phosphodiesterase 1, Phosphodiesterase 1A (PDE1A), Phosphodiesterase 1C (PDE1C), Phosphodiesterase 3 (PDE3), Phosphodiesterase 7, Phosphodiesterase 8, cAMP-specific 3',5'-cyclic phosphodiesterase 4A, cAMP-specific 3',5'-cyclic phosphodiesterase 4B, cAMP-specific 3',5'-cyclic phosphodiesterase 4C, cAMP-specific 3',5'-cyclic phosphodiesterase 4D, cAMP-specific 3',5'-cyclic phosphodiesterase 7B, cGMP-inhibited 3',5'-cyclic phosphodiesterase B, and cGMP-specific 3',5'-cyclic phosphodiesterase, Pfizer Global Research and Development, Affinity

12 Research products, page 1 of 2

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